Pérez, Oswaldo; Schipper, Nicolaas; Bollmark, Martin
(American Chemical Society, 2021-10-19)
Cyclic guanosine monophosphorothioate analogue 1a is currently showing potential as a drug for the treatment of inherited retinal neurodegenerations. To support ongoing preclinical and clinical work, we have developed a diastereoselective synthesis via ...